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GRK2 and GNAQ
Number of citations of the paper that reports this interaction (PubMedID
12885252
)
0
Data Source:
HPRD
(in vivo, in vitro)
GRK2
GNAQ
Description
G protein-coupled receptor kinase 2
G protein subunit alpha q
Image
GO Annotations
Cellular Component
Cytoplasm
Cytosol
Plasma Membrane
Cilium
Membrane
Cytoplasmic Side Of Mitochondrial Outer Membrane
Cell Projection
Synapse
Presynapse
Postsynapse
Photoreceptor Outer Segment
Nucleus
Cytoplasm
Lysosomal Membrane
Golgi Apparatus
Heterotrimeric G-protein Complex
Plasma Membrane
Membrane
Nuclear Membrane
Extracellular Exosome
Postsynaptic Cytosol
Molecular Function
Nucleotide Binding
G Protein-coupled Receptor Binding
Protein Kinase Activity
Protein Serine/threonine Kinase Activity
G Protein-coupled Receptor Kinase Activity
Protein Binding
ATP Binding
Kinase Activity
Transferase Activity
Alpha-2A Adrenergic Receptor Binding
Edg-2 Lysophosphatidic Acid Receptor Binding
Beta-adrenergic Receptor Kinase Activity
Nucleotide Binding
G Protein-coupled Receptor Binding
GTPase Activity
G Protein Activity
GTPase Activator Activity
Protein Binding
GTP Binding
Hydrolase Activity
Guanyl Nucleotide Binding
Enzyme Regulator Activity
G-protein Beta/gamma-subunit Complex Binding
Metal Ion Binding
Biological Process
Regulation Of The Force Of Heart Contraction
Desensitization Of G Protein-coupled Receptor Signaling Pathway
Negative Regulation Of The Force Of Heart Contraction By Chemical Signal
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Acetylcholine Receptor Signaling Pathway
Tachykinin Receptor Signaling Pathway
Heart Development
Viral Genome Replication
Receptor Internalization
Positive Regulation Of Catecholamine Secretion
Negative Regulation Of Striated Muscle Contraction
Symbiont Entry Into Host Cell
Cardiac Muscle Contraction
Negative Regulation Of Relaxation Of Smooth Muscle
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
Adenylate Cyclase-activating G Protein-coupled Receptor Signaling Pathway
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Phospholipase C-activating G Protein-coupled Glutamate Receptor Signaling Pathway
Phospholipase C-activating Serotonin Receptor Signaling Pathway
G Protein-coupled Acetylcholine Receptor Signaling Pathway
Glutamate Receptor Signaling Pathway
Neuropeptide Signaling Pathway
Blood Coagulation
Phototransduction, Visible Light
Entrainment Of Circadian Clock
Hormone-mediated Signaling Pathway
Regulation Of Platelet Activation
Response To Prostaglandin E
Protein Stabilization
Regulation Of Canonical Wnt Signaling Pathway
Cellular Response To Acidic PH
Adenylate Cyclase-activating G Protein-coupled CAMP Receptor Signaling Pathway
Pathways
Calmodulin induced events
G alpha (q) signalling events
G alpha (s) signalling events
Activation of SMO
Activation of SMO
Cargo recognition for clathrin-mediated endocytosis
PLC beta mediated events
PLC beta mediated events
G-protein activation
Acetylcholine regulates insulin secretion
Acetylcholine regulates insulin secretion
G alpha (q) signalling events
G alpha (q) signalling events
ADP signalling through P2Y purinoceptor 1
ADP signalling through P2Y purinoceptor 1
Thromboxane signalling through TP receptor
Fatty Acids bound to GPR40 (FFAR1) regulate insulin secretion
Fatty Acids bound to GPR40 (FFAR1) regulate insulin secretion
Thrombin signalling through proteinase activated receptors (PARs)
Cooperation of PDCL (PhLP1) and TRiC/CCT in G-protein beta folding
High laminar flow shear stress activates signaling by PIEZO1 and PECAM1:CDH5:KDR in endothelial cells
Turbulent (oscillatory, disturbed) flow shear stress activates signaling by PIEZO1 and integrins in endothelial cells
Drugs
ATP
Diseases
GWAS
Bipolar disorder (
31043756
)
Electrocardiogram morphology (amplitude at temporal datapoints) (
32916098
)
Interacting Genes
49 interacting genes:
ADRA2A
ADRB2
AGTR1
AKAP12
ARRB1
BDKRB2
CAPN2
CAV1
CCR4
CCR5
CSNK2B
EGF
EGFR
EPHA2
ERBB2
FBXO25
FPR1
FSHR
GIT1
GIT2
GNA15
GNAQ
GNB3
GRM1
HDAC6
KCNIP3
MAPK3
MC4R
MDM2
NCS1
OPRD1
PDC
PDCL
PDE6G
PEBP1
PIK3CG
PLCB1
PRKACA
PRKCA
PRKCB
PRKCD
PRKCG
RASGRF1
RCVRN
RHO
RPLP2
SNCA
SRC
TPM2
48 interacting genes:
ADHFE1
ADRA1B
AIP
AKAP13
BDKRB1
BTK
CCR5
CHRM3
CRHR1
CYTH1
CYTH2
FFAR1
FFAR2
GALR2
GRK2
GRM2
GRM4
GRM7
HTR2A
HTR2B
HTR2C
HTR6
KDR
LUM
MRGPRX1
NHERF1
NT5C3A
PIK3CA
PLCB1
PLCB2
PPT1
PTGIR
RGS13
RGS16
RGS18
RGS2
RGS4
RGS5
RGS7
RIC8A
RIC8B
S1PR2
S1PR3
TBXA2R
TSHR
TTC1
TUB
VIPR1
Entrez ID
156
2776
HPRD ID
00182
02998
Ensembl ID
ENSG00000173020
ENSG00000156052
Uniprot IDs
A0A0S2Z392
P25098
A0A024R240
P50148
PDB IDs
1BAK
3CIK
3KRW
3KRX
3V5W
4MK0
4PNK
5HE1
5UKK
5UKL
5UUU
5UVC
5WG3
5WG4
5WG5
6C2Y
6U7C
7K7L
7K7Z
7PWD
6VU5
7EZM
7F6G
7F6H
7F6I
7F8W
7W3Z
7W40
7XOW
8G59
8IA7
8IYS
8J9N
8JPB
8JPC
8JPE
8SZG
8UQN
8UQO
8XGO
8XGS
8Y52
8ZJD
8ZJE
9K27
Enriched GO Terms of Interacting Partners
?
G Protein-coupled Receptor Signaling Pathway
Regulation Of Cell Communication
Signal Transduction
Regulation Of Signaling
Regulation Of Signal Transduction
Regulation Of MAPK Cascade
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of Intracellular Signal Transduction
Positive Regulation Of MAPK Cascade
Plasma Membrane
Regulation Of Biological Quality
Positive Regulation Of Intracellular Signal Transduction
Positive Regulation Of Cell Communication
Positive Regulation Of Signaling
System Process
Positive Regulation Of Signal Transduction
Regulation Of G Protein-coupled Receptor Signaling Pathway
Regulation Of Multicellular Organismal Process
Modulation Of Chemical Synaptic Transmission
Enzyme Binding
Intracellular Signal Transduction
G Protein-coupled Receptor Activity
Regulation Of Transport
Epidermal Growth Factor Receptor Signaling Pathway
Intracellular Signaling Cassette
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
ERBB Signaling Pathway
Regulation Of Vesicle-mediated Transport
Response To Lipid
Cell Surface Receptor Signaling Pathway
ERBB2 Signaling Pathway
Nervous System Process
Response To Hormone
Response To Growth Factor
Calcium,diacylglycerol-dependent Serine/threonine Kinase Activity
Regulation Of Locomotion
Positive Regulation Of Protein Localization
Regulation Of System Process
Positive Regulation Of Cell Migration
Cell Surface Receptor Protein Tyrosine Kinase Signaling Pathway
Regulation Of Metal Ion Transport
Regulation Of Phosphorus Metabolic Process
Regulation Of Cellular Component Organization
Positive Regulation Of Cell Motility
Positive Regulation Of Locomotion
Protein Kinase C Signaling
Negative Regulation Of Catabolic Process
Cellular Response To Oxygen-containing Compound
Regulation Of ERK1 And ERK2 Cascade
Regulation Of Proteolysis
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Activity
Signal Transduction
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
Plasma Membrane
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of Cell Communication
Regulation Of Signaling
Adenylate Cyclase-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Signaling Pathway, Coupled To Cyclic Nucleotide Second Messenger
G-protein Alpha-subunit Binding
Regulation Of Signal Transduction
Positive Regulation Of Cytosolic Calcium Ion Concentration
Regulation Of Biological Quality
System Process
Serotonin Receptor Signaling Pathway
Release Of Sequestered Calcium Ion Into Cytosol
Negative Regulation Of Sequestering Of Calcium Ion
Positive Regulation Of Phosphatidylinositol Biosynthetic Process
Gq/11-coupled Serotonin Receptor Activity
Serotonin Receptor Activity
Membrane
G Protein-coupled Serotonin Receptor Activity
Cell-cell Signaling
Regulation Of Amine Transport
Regulation Of Sequestering Of Calcium Ion
G Protein-coupled Serotonin Receptor Complex
Signaling
Adenylate Cyclase-inhibiting G Protein-coupled Receptor Signaling Pathway
Neurotransmitter Receptor Activity
Cell Communication
Calcium Ion Transmembrane Import Into Cytosol
Regulation Of System Process
G Protein-coupled Serotonin Receptor Signaling Pathway
Negative Regulation Of G Protein-coupled Receptor Signaling Pathway
Muscle System Process
GTPase Activator Activity
Phosphatidylinositol-4,5-bisphosphate Phospholipase C Activity
Regulation Of Transport
Positive Regulation Of Cell Communication
Positive Regulation Of Signaling
Regulation Of Secretion
Phospholipase C-activating Serotonin Receptor Signaling Pathway
Muscle Contraction
Adenylate Cyclase-inhibiting G Protein-coupled Glutamate Receptor Signaling Pathway
Chemical Synaptic Transmission
Serotonin Binding
Guanyl-nucleotide Exchange Factor Activity
Regulation Of Secretion By Cell
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