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GRK6 and EDNRB
Number of citations of the paper that reports this interaction (PubMedID
9211925
)
0
Data Source:
HPRD
(in vitro)
GRK6
EDNRB
Description
G protein-coupled receptor kinase 6
endothelin receptor type B
Image
GO Annotations
Cellular Component
Cytoplasm
Plasma Membrane
Membrane
Plasma Membrane
Membrane
Nuclear Membrane
Molecular Function
Nucleotide Binding
Protein Kinase Activity
Protein Serine/threonine Kinase Activity
G Protein-coupled Receptor Kinase Activity
Protein Binding
ATP Binding
Kinase Activity
Transferase Activity
Beta-adrenergic Receptor Kinase Activity
G Protein-coupled Receptor Activity
Endothelin Receptor Activity
Protein Binding
Peptide Hormone Binding
Type 1 Angiotensin Receptor Binding
Biological Process
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
Regulation Of G Protein-coupled Receptor Signaling Pathway
Regulation Of Signal Transduction
Wnt Signaling Pathway
Negative Regulation Of Transcription By RNA Polymerase II
Neural Crest Cell Migration
Renin Secretion Into Blood Stream
Regulation Of Heart Rate
Regulation Of PH
Signal Transduction
Cell Surface Receptor Signaling Pathway
G Protein-coupled Receptor Signaling Pathway
Negative Regulation Of Adenylate Cyclase Activity
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Positive Regulation Of Cytosolic Calcium Ion Concentration
Nervous System Development
Peripheral Nervous System Development
Posterior Midgut Development
Regulation Of Blood Pressure
Positive Regulation Of Cell Population Proliferation
Gene Expression
Negative Regulation Of Neuron Maturation
Vein Smooth Muscle Contraction
Vascular Associated Smooth Muscle Contraction
Calcium-mediated Signaling
CGMP-mediated Signaling
Heparin Proteoglycan Metabolic Process
Melanocyte Differentiation
Regulation Of Fever Generation
Aldosterone Metabolic Process
Response To Lipopolysaccharide
Enteric Smooth Muscle Cell Differentiation
Positive Regulation Of Urine Volume
Renal Sodium Excretion
Epithelial Fluid Transport
Vasoconstriction
Vasodilation
Negative Regulation Of Apoptotic Process
Positive Regulation Of Canonical NF-kappaB Signal Transduction
Pigmentation
Developmental Pigmentation
Macrophage Chemotaxis
Response To Pain
Enteric Nervous System Development
Regulation Of Epithelial Cell Proliferation
Negative Regulation Of Protein Metabolic Process
Sodium Ion Homeostasis
Canonical Wnt Signaling Pathway
Positive Regulation Of Penile Erection
Establishment Of Endothelial Barrier
Renal Sodium Ion Absorption
Calcium Ion Transmembrane Transport
Cellular Response To Lipopolysaccharide
Protein Transmembrane Transport
Podocyte Differentiation
Endothelin Receptor Signaling Pathway
Renal Albumin Absorption
Neuroblast Migration
Chordate Pharynx Development
Response To Sodium Phosphate
Response To Endothelin
Pathways
G alpha (s) signalling events
Peptide ligand-binding receptors
G alpha (q) signalling events
Transcriptional and post-translational regulation of MITF-M expression and activity
Drugs
Bosentan
IRL-1620
Sitaxentan
Ambrisentan
Enrasentan
Tezosentan
Macitentan
Diseases
Hirschsprung disease (HD)
Waardenburg syndrome (WS)
ABCD syndrome
Nasopharyngeal cancer
GWAS
Activated partial thromboplastin time (
22703881
)
Cardiac troponin-I levels (
31014085
)
Chronic kidney disease (
20383146
)
Extremely high intelligence (
29520040
)
Glycine levels (
30837465
)
Intelligence (MTAG) (
29326435
)
Metabolite levels (
22916037
)
Neutrophil percentage of white cells (
32888494
)
Tinnitus (
33742053
)
Waist-to-hip ratio adjusted for BMI (
26426971
)
Waist-to-hip ratio adjusted for BMI (age <50) (
26426971
)
Waist-to-hip ratio adjusted for BMI x sex x age interaction (4df test) (
26426971
)
Appendicular lean mass (
33097823
)
Craniofacial microsomia (
26853712
)
Hair color (
23548203
29662168
)
Total ventricular volume (Alzheimer's disease interaction) (
21116278
)
Interacting Genes
19 interacting genes:
ADRB2
BDKRB2
CHRM3
EDNRA
EDNRB
FBXO7
FSHR
GIT1
ITGA5
KCNIP3
LTB4R
NHERF1
PRSS23
RCVRN
RHO
SNCA
SNCB
SNCG
TBXA2R
7 interacting genes:
CAV1
EDN1
EDN3
GNA11
GNA13
GRK6
NOS3
Entrez ID
2870
1910
HPRD ID
02925
08834
Ensembl ID
ENSG00000198055
ENSG00000136160
Uniprot IDs
B3KPS5
P43250
P24530
PDB IDs
2ACX
3NYN
3NYO
5GLH
5GLI
5X93
5XPR
6IGK
6IGL
6LRY
8HBD
8HCX
8IY5
8IY6
8XGR
8XVE
8XVH
8XWP
8XWQ
8ZRT
Enriched GO Terms of Interacting Partners
?
Smooth Muscle Contraction
G Protein-coupled Receptor Activity
Muscle Contraction
G Protein-coupled Receptor Signaling Pathway
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
System Process
Muscle System Process
Cuprous Ion Binding
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
Vascular Process In Circulatory System
Blood Vessel Diameter Maintenance
Regulation Of Tube Size
Regulation Of Cell Communication
Regulation Of Signaling
Regulation Of Blood Pressure
Circulatory System Process
Endothelin Receptor Activity
Regulation Of System Process
Renal Sodium Ion Transport
Phosphatidylinositol-4,5-bisphosphate Phospholipase C Activity
Regulation Of Platelet-derived Growth Factor Receptor Signaling Pathway
Regulation Of Monoatomic Ion Transport
Vasoconstriction
Renal Albumin Absorption
Regulation Of Multicellular Organismal Process
Signal Transduction
Synaptic Vesicle Endocytosis
Type 1 Angiotensin Receptor Binding
Regulation Of Signal Transduction
Secretion
Renal Absorption
Catecholamine Metabolic Process
Presynaptic Endocytosis
Regulation Of Transport
Positive Regulation Of Cytosolic Calcium Ion Concentration
Regulation Of Biological Quality
Adenylate Cyclase-activating G Protein-coupled Receptor Signaling Pathway
Renal Protein Absorption
Vasodilation
Regulation Of Metal Ion Transport
Axon Terminus
Regulation Of Smooth Muscle Contraction
Locomotory Behavior
Biogenic Amine Metabolic Process
Cellular Response To Follicle-stimulating Hormone Stimulus
Heparin Proteoglycan Metabolic Process
Enteric Nervous System Development
Endothelin Receptor Signaling Pathway
Podocyte Differentiation
Amine Metabolic Process
Regulation Of Systemic Arterial Blood Pressure By Endothelin
Regulation Of Blood Pressure
Regulation Of Systemic Arterial Blood Pressure Mediated By A Chemical Signal
Blood Vessel Diameter Maintenance
Vasoconstriction
Regulation Of Tube Size
Endothelin B Receptor Binding
Regulation Of Systemic Arterial Blood Pressure
Vein Smooth Muscle Contraction
Regulation Of Heart Contraction
Regulation Of Locomotion
Regulation Of Smooth Muscle Contraction
Regulation Of Vasoconstriction
Regulation Of Muscle System Process
Regulation Of The Force Of Heart Contraction By Chemical Signal
Regulation Of Blood Circulation
Regulation Of Blood Coagulation
Vascular Process In Circulatory System
Regulation Of Hemostasis
Regulation Of Potassium Ion Transport
Regulation Of Developmental Process
Circulatory System Process
Artery Smooth Muscle Contraction
G Protein-coupled Receptor Signaling Pathway
Tonic Smooth Muscle Contraction
Regulation Of Heart Rate
Endothelin Receptor Signaling Pathway
Positive Regulation Of Cation Transmembrane Transport
Positive Regulation Of Monoatomic Ion Transmembrane Transport
Regulation Of Monoatomic Ion Transport
Vascular Associated Smooth Muscle Contraction
Guanyl Nucleotide Binding
Regulation Of Wound Healing
Regulation Of Cell Migration
Positive Regulation Of Hormone Secretion
Regulation Of Cell Motility
Nitric Oxide Biosynthetic Process
G-protein Beta/gamma-subunit Complex Binding
Regulation Of Muscle Contraction
Regulation Of Response To Wounding
Regulation Of The Force Of Heart Contraction
Positive Regulation Of Monoatomic Ion Transport
Positive Regulation Of Cell Migration
Regulation Of System Process
Intracellular Calcium Ion Homeostasis
Positive Regulation Of Heart Rate
Negative Regulation Of Potassium Ion Transport
Positive Regulation Of Cell Motility
Nitric Oxide Metabolic Process
Positive Regulation Of Smooth Muscle Contraction
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Tagcloud (Intersection)
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