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HTR2C and ARRB2
Number of citations of the paper that reports this interaction (PubMedID
18768750
)
52
Data Source:
HPRD
(in vivo)
HTR2C
ARRB2
Description
5-hydroxytryptamine receptor 2C
arrestin beta 2
Image
No pdb structure
GO Annotations
Cellular Component
Plasma Membrane
Membrane
Dendrite
Synapse
G Protein-coupled Serotonin Receptor Complex
Nucleus
Nucleoplasm
Cytoplasm
Cytosol
Plasma Membrane
Clathrin-coated Pit
Membrane
Endocytic Vesicle
Endocytic Vesicle Membrane
Cytoplasmic Vesicle
Postsynapse
Glutamatergic Synapse
Molecular Function
Gq/11-coupled Serotonin Receptor Activity
G Protein-coupled Receptor Activity
G Protein-coupled Serotonin Receptor Activity
Protein Binding
Neurotransmitter Receptor Activity
Identical Protein Binding
Serotonin Binding
1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine Binding
Serotonin Receptor Activity
G Protein-coupled Receptor Binding
Signaling Receptor Binding
Protein Binding
Enzyme Binding
Protein-macromolecule Adaptor Activity
Ubiquitin Protein Ligase Binding
Angiotensin Receptor Binding
D1 Dopamine Receptor Binding
Protein Kinase B Binding
Molecular Adaptor Activity
Biological Process
Behavioral Fear Response
Intracellular Calcium Ion Homeostasis
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Signaling Pathway, Coupled To Cyclic Nucleotide Second Messenger
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Phospholipase C-activating Serotonin Receptor Signaling Pathway
Serotonin Receptor Signaling Pathway
Chemical Synaptic Transmission
Locomotory Behavior
Feeding Behavior
Positive Regulation Of Phosphatidylinositol Biosynthetic Process
CGMP-mediated Signaling
Regulation Of Nervous System Process
Regulation Of Appetite
Regulation Of Corticotropin-releasing Hormone Secretion
Positive Regulation Of Fat Cell Differentiation
Positive Regulation Of Calcium-mediated Signaling
Release Of Sequestered Calcium Ion Into Cytosol
Positive Regulation Of ERK1 And ERK2 Cascade
G Protein-coupled Serotonin Receptor Signaling Pathway
Desensitization Of G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Internalization
Positive Regulation Of Receptor Internalization
Transcription By RNA Polymerase II
Signal Transduction
Transforming Growth Factor Beta Receptor Signaling Pathway
Canonical NF-kappaB Signal Transduction
Adult Walking Behavior
Regulation Of G Protein-coupled Receptor Signaling Pathway
Negative Regulation Of Signal Transduction
Positive Regulation Of Cardiac Muscle Hypertrophy
Positive Regulation Of Gene Expression
Protein Transport
Protein Ubiquitination
Sensory Perception Of Pain
Negative Regulation Of Protein Ubiquitination
Receptor Internalization
Negative Regulation Of NF-kappaB Transcription Factor Activity
Positive Regulation Of Synaptic Transmission, Dopaminergic
Negative Regulation Of Interleukin-1 Beta Production
Negative Regulation Of Interleukin-12 Production
Negative Regulation Of Interleukin-6 Production
Negative Regulation Of Tumor Necrosis Factor Production
Negative Regulation Of Toll-like Receptor Signaling Pathway
Negative Regulation Of Canonical NF-kappaB Signal Transduction
Proteasome-mediated Ubiquitin-dependent Protein Catabolic Process
Negative Regulation Of Natural Killer Cell Mediated Cytotoxicity
Modulation Of Chemical Synaptic Transmission
Positive Regulation Of Phosphatidylinositol 3-kinase/protein Kinase B Signal Transduction
Negative Regulation Of Phosphatidylinositol 3-kinase/protein Kinase B Signal Transduction
Excitatory Postsynaptic Potential
Cell Chemotaxis
Positive Regulation Of ERK1 And ERK2 Cascade
Postsynaptic Signal Transduction
Beta-arrestin-dependent Dopamine Receptor Signaling Pathway
Positive Regulation Of Intracellular Signal Transduction
Positive Regulation Of Cardiac Muscle Cell Differentiation
Pathways
Serotonin receptors
G alpha (q) signalling events
Activated NOTCH1 Transmits Signal to the Nucleus
G alpha (s) signalling events
Thrombin signalling through proteinase activated receptors (PARs)
WNT5A-dependent internalization of FZD4
Activation of SMO
Activation of SMO
MAP2K and MAPK activation
Ub-specific processing proteases
Signaling by moderate kinase activity BRAF mutants
Signaling by high-kinase activity BRAF mutants
Signaling by BRAF and RAF1 fusions
Paradoxical activation of RAF signaling by kinase inactive BRAF
Cargo recognition for clathrin-mediated endocytosis
Clathrin-mediated endocytosis
Signaling downstream of RAS mutants
Signaling by RAF1 mutants
TGFBR3 regulates TGF-beta signaling
Drugs
Tramadol
Ziprasidone
Methysergide
Cabergoline
Dihydroergotamine
Amitriptyline
Olanzapine
Clozapine
Mirtazapine
Loxapine
Promazine
Cyproheptadine
Imipramine
Fluoxetine
Chlorpromazine
Chlorpromazine
Haloperidol
Nortriptyline
Amoxapine
Fenfluramine
Lisuride
Fluphenazine
Trazodone
Ergotamine
Apomorphine
Paroxetine
Trimipramine
Risperidone
Propiomazine
Minaprine
Flupentixol
Cyclobenzaprine
Maprotiline
Ergoloid mesylate
Tegaserod
Doxepin
Nefazodone
Desipramine
Escitalopram
Pergolide
Dexfenfluramine
Bromocriptine
Ketamine
Quetiapine
Aripiprazole
Chlorprothixene
Clomipramine
Paliperidone
Yohimbine
Methotrimeprazine
Midomafetamine
4-Bromo-2,5-dimethoxyphenethylamine
Lorcaserin
Dapoxetine
Lofexidine
Pimavanserin
Epicept NP-1
Cariprazine
Sertindole
Mianserin
Pizotifen
Asenapine
Ocaperidone
Dotarizine
Deramciclane
Agomelatine
Esmirtazapine
Nandrolone decanoate
Captodiame
Viloxazine
Etoperidone
Lorpiprazole
Setiptiline
Dihydroergocornine
m-Chlorophenylpiperazine
Gilteritinib
Sarpogrelate
Eplivanserin
Tiapride
Dihydroergocristine
2,5-Dimethoxy-4-ethylthioamphetamine
Aripiprazole lauroxil
Diseases
GWAS
Behcet's disease (
33393726
)
Lymphocyte count (
27863252
32888494
)
Lymphocyte percentage of white cells (
32888494
)
White blood cell count (
32888494
)
Interacting Genes
34 interacting genes:
APBA1
ARLN
ARRB2
ATP2B3
ATP6AP2
ATP6V0C
CALM1
CBX3
CNIH1
CRELD1
DLG4
EMP1
ERG28
GHITM
GJA1
GNAQ
GPR37
GPRC5B
LIN7C
MPDZ
PLP1
RTN4
SGCB
SLC29A1
SLC39A1
SLC39A9
SLC71A1
SNTA1
SPNS1
TM9SF2
TMBIM6
TMEM147
TMEM94
TPI1
60 interacting genes:
ADRB2
AGTR1
AGTR2
AP1B1
AP2M1
ARF6
AVPR2
BCAS1
C5AR1
CDC42
CLTC
CRHR1
CSNK2A1
CSNK2A2
CXCR4
CYTH2
DLG4
DVL2
EGFR
EIF2AK4
FLNA
FZD4
HCRTR1
HIPK3
HTR2C
ITCH
LHCGR
LIMK1
MAP2K4
MAP3K5
MAPK1
MAPK10
MAPK9
MAS1
MDM2
MED8
NDUFS7
NEDD4L
NFKBIA
NTS
NTSR1
OPRD1
OXER1
OXTR
PDE4D
PTAFR
PTGDS
RAF1
RALGDS
RHO
SLC9A5
SMARCC2
SNCA
STC2
SUMO1
SUMO2
TGFBR3
TRH
UBC
UBE2I
Entrez ID
3358
409
HPRD ID
02429
00147
Ensembl ID
ENSG00000147246
ENSG00000141480
Uniprot IDs
K9J958
P28335
K7ENA6
P32121
Q59EM5
Q68DZ5
PDB IDs
6BQG
6BQH
8DPF
8DPG
8DPH
8DPI
8ZMF
Enriched GO Terms of Interacting Partners
?
Membrane
Endoplasmic Reticulum Membrane
Plasma Membrane
Transmembrane Transport
Cellular Homeostasis
Intracellular Chemical Homeostasis
Homeostatic Process
Chemical Homeostasis
Synapse
Monoatomic Ion Transmembrane Transport
Intracellular Monoatomic Cation Homeostasis
Intracellular Monoatomic Ion Homeostasis
Inorganic Cation Transmembrane Transport
Endoplasmic Reticulum
PDZ Domain Binding
Monoatomic Cation Transmembrane Transport
Ubiquitin Protein Ligase Binding
Monoatomic Cation Homeostasis
Regulation Of Lysosomal Lumen PH
Monoatomic Ion Homeostasis
Inorganic Ion Transmembrane Transport
Monoatomic Ion Transport
D1 Dopamine Receptor Binding
Monoatomic Cation Transport
Glutamatergic Synapse
Golgi Lumen Acidification
Vacuolar Proton-transporting V-type ATPase, V0 Domain
Regulation Of Membrane Potential
Neuron Cellular Homeostasis
Glutamate Secretion
Endosomal Lumen Acidification
G Protein-coupled Receptor Binding
Dystrophin-associated Glycoprotein Complex
Proton-transporting V-type ATPase Complex
Synaptic Vesicle Lumen Acidification
Regulation Of Intracellular PH
Bounding Membrane Of Organelle
Regulation Of Cellular PH
Regulation Of System Process
Metal Ion Transmembrane Transporter Activity
Protein-macromolecule Adaptor Activity
Regulation Of Biological Quality
Metal Ion Transport
Regulation Of PH
Zinc Ion Transmembrane Transporter Activity
Positive Regulation Of Macrophage Cytokine Production
Postsynapse
Lysosomal Lumen Acidification
Anchoring Junction
Zinc Ion Transmembrane Transport
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Activity
Plasma Membrane
Signal Transduction
Regulation Of Biological Quality
Regulation Of Cell Communication
Regulation Of Signaling
Regulation Of Signal Transduction
Positive Regulation Of Cell Communication
Positive Regulation Of Signaling
Cell Surface Receptor Signaling Pathway
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
Regulation Of Intracellular Signal Transduction
Intracellular Signaling Cassette
Regulation Of Multicellular Organismal Process
Protein Serine Kinase Activity
Regulation Of Systemic Arterial Blood Pressure Mediated By A Chemical Signal
Positive Regulation Of Metabolic Process
Regulation Of Protein Catabolic Process
Intracellular Signal Transduction
Protein Serine/threonine Kinase Activity
Protein Kinase Activity
Clathrin-coated Endocytic Vesicle Membrane
Angiotensin Type II Receptor Activity
Regulation Of Transport
Positive Regulation Of Signal Transduction
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of Cellular Component Organization
Regulation Of Metal Ion Transport
Regulation Of MAPK Cascade
Regulation Of System Process
Regulation Of Systemic Arterial Blood Pressure
Glutamatergic Synapse
Regulation Of Developmental Process
Positive Regulation Of Locomotion
Negative Regulation Of Systemic Arterial Blood Pressure
Ubiquitin Protein Ligase Binding
Enzyme Binding
Blood Vessel Diameter Maintenance
Regulation Of Tube Size
Kinase Activity
Import Into Cell
Postsynapse
Regulation Of Monoatomic Ion Transport
Response To Stress
Regulation Of Blood Pressure
Neuron Spine
Positive Regulation Of Neuron Projection Arborization
Endocytosis
Positive Regulation Of Cell Migration
Tagcloud
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Tagcloud (Difference)
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Tagcloud (Intersection)
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