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CCR5 and GRK3
Number of citations of the paper that reports this interaction (PubMedID
10085131
)
0
Data Source:
HPRD
(in vitro)
CCR5
GRK3
Description
C-C motif chemokine receptor 5
G protein-coupled receptor kinase 3
Image
No pdb structure
GO Annotations
Cellular Component
Cytoplasm
Endosome
Plasma Membrane
External Side Of Plasma Membrane
Cell Surface
Membrane
Cytoplasm
Cytosol
Plasma Membrane
Cell Projection
Synapse
Presynapse
Postsynapse
Molecular Function
Virus Receptor Activity
Actin Binding
Phosphatidylinositol-4,5-bisphosphate Phospholipase C Activity
G Protein-coupled Receptor Activity
Chemokine Receptor Activity
Protein Binding
Coreceptor Activity
C-C Chemokine Receptor Activity
C-C Chemokine Binding
Identical Protein Binding
Chemokine (C-C Motif) Ligand 5 Binding
Nucleotide Binding
G Protein-coupled Receptor Binding
Protein Kinase Activity
Protein Serine/threonine Kinase Activity
G Protein-coupled Receptor Kinase Activity
Protein Binding
ATP Binding
Kinase Activity
Transferase Activity
Beta-adrenergic Receptor Kinase Activity
Biological Process
MAPK Cascade
Dendritic Cell Chemotaxis
Calcium Ion Transport
Apoptotic Process
Chemotaxis
Defense Response
Inflammatory Response
Immune Response
Cellular Defense Response
Signal Transduction
Cell Surface Receptor Signaling Pathway
G Protein-coupled Receptor Signaling Pathway
Positive Regulation Of Cytosolic Calcium Ion Concentration
Cell-cell Signaling
Release Of Sequestered Calcium Ion Into Cytosol By Sarcoplasmic Reticulum
Calcium-mediated Signaling
Signaling
Symbiont Entry Into Host Cell
Cell Chemotaxis
Chemokine-mediated Signaling Pathway
Response To Cholesterol
Cellular Response To Lipopolysaccharide
Cellular Response To Cytokine Stimulus
Negative Regulation Of Macrophage Apoptotic Process
Desensitization Of G Protein-coupled Receptor Signaling Pathway
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
Receptor Internalization
Pathways
Binding and entry of HIV virion
Chemokine receptors bind chemokines
G alpha (i) signalling events
Interleukin-10 signaling
G alpha (s) signalling events
Cargo recognition for clathrin-mediated endocytosis
Drugs
Maraviroc
AMD-070
CCR5 mAb
Leronlimab
Aplaviroc
Vicriviroc
Ibalizumab
INCB-9471
ATP
Diseases
GWAS
Blood protein levels in cardiovascular risk (
28369058
)
Celiac disease (
20190752
)
Cerebrospinal fluid levels of Alzheimer's disease-related proteins (
25340798
)
Granulocyte percentage of myeloid white cells (
27863252
)
Inflammatory bowel disease (
26192919
)
Type 1 diabetes (
25751624
)
Ulcerative colitis (
26192919
28067908
)
Interacting Genes
43 interacting genes:
AFP
ARL6IP5
ARRB1
CCL11
CCL13
CCL14
CCL16
CCL2
CCL3
CCL3L1
CCL3L3
CCL4
CCL5
CCL7
CCL8
CD4
CST9L
CTBP2
CXCR4
DNM2
EMP1
ETV5
GNAI1
GNAI2
GNAI3
GNAO1
GNAQ
GRK2
GRK3
IL24
JAK1
JAK2
LCK
ORM1
PRAF2
PSMA5
PTK2
PTK2B
SLC20A2
STAT1
STAT3
STAT5A
TXK
11 interacting genes:
ADRB2
AGTR1
BDKRB2
CCR4
CCR5
CXCR4
GIT1
HSPB1
OPRM1
SMURF1
SNCA
Entrez ID
1234
157
HPRD ID
03223
00183
Ensembl ID
ENSG00000160791
ENSG00000100077
Uniprot IDs
P51681
Q38L21
P35626
Q8N433
PDB IDs
2L87
2MZX
2RLL
2RRS
4MBS
5UIW
5YD3
5YD4
5YD5
5YY4
6FGP
6MEO
6MET
7F1Q
7F1R
7F1S
7NJZ
7NW3
7O7F
8AS2
8AS3
Enriched GO Terms of Interacting Partners
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Chemokine-mediated Signaling Pathway
CCR Chemokine Receptor Binding
Cytokine-mediated Signaling Pathway
Chemokine Activity
G Protein-coupled Receptor Signaling Pathway
Eosinophil Chemotaxis
Eosinophil Migration
Positive Regulation Of Cell Migration
Positive Regulation Of Cell Motility
Positive Regulation Of Locomotion
Antimicrobial Humoral Response
Antimicrobial Humoral Immune Response Mediated By Antimicrobial Peptide
Cell Chemotaxis
Cytokine Activity
CCR5 Chemokine Receptor Binding
Immune System Process
Immune Response
Cell Surface Receptor Signaling Pathway
Regulation Of Cell Migration
Humoral Immune Response
Regulation Of Cell Motility
Signal Transduction
Regulation Of Locomotion
Granulocyte Chemotaxis
Leukocyte Migration
Chemotaxis
Granulocyte Migration
Defense Response
Cell Migration
Leukocyte Chemotaxis
Inflammatory Response
Locomotion
Response To Other Organism
Response To External Biotic Stimulus
Cell Motility
Regulation Of Lymphocyte Chemotaxis
Myeloid Leukocyte Migration
Defense Response To Symbiont
Positive Regulation Of Natural Killer Cell Chemotaxis
Defense Response To Other Organism
Guanyl Nucleotide Binding
CCR1 Chemokine Receptor Binding
G Protein-coupled Receptor Binding
Positive Regulation Of Multicellular Organismal Process
Positive Regulation Of Lymphocyte Chemotaxis
Cell Surface Receptor Signaling Pathway Via STAT
Non-membrane Spanning Protein Tyrosine Kinase Activity
G-protein Beta/gamma-subunit Complex Binding
Protein Kinase Activity
Interleukin-9-mediated Signaling Pathway
G Protein-coupled Receptor Activity
Positive Regulation Of Cytosolic Calcium Ion Concentration
G Protein-coupled Receptor Signaling Pathway
Regulation Of Biological Quality
Chemokine Receptor Activity
C-C Chemokine Binding
C-C Chemokine Receptor Activity
Negative Regulation Of Cell Communication
Negative Regulation Of Signaling
Signal Transduction
Regulation Of Cell Communication
Regulation Of Signaling
Calcium-mediated Signaling
Endosome
Cell Surface Receptor Signaling Pathway
Cell Chemotaxis
Negative Regulation Of Signal Transduction
Regulation Of Multicellular Organismal Process
Inflammatory Response
Regulation Of Signal Transduction
Chemokine-mediated Signaling Pathway
Positive Regulation Of Catabolic Process
Response To Stress
Plasma Membrane
Chemotaxis
Dendritic Cell Chemotaxis
Intracellular Signal Transduction
Symbiont Entry Into Host Cell
Locomotion
Regulation Of Autophagy
Phosphatidylinositol-4,5-bisphosphate Phospholipase C Activity
Dendritic Cell Migration
Positive Regulation Of Developmental Process
Blood Vessel Diameter Maintenance
Regulation Of G Protein-coupled Receptor Signaling Pathway
Regulation Of Tube Size
Biological Process Involved In Interaction With Host
Regulation Of Systemic Arterial Blood Pressure Mediated By A Chemical Signal
Positive Regulation Of Organelle Organization
Regulation Of Systemic Arterial Blood Pressure
Response To Cytokine
Positive Regulation Of Cellular Component Organization
Positive Regulation Of Metabolic Process
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
Vasodilation
Negative Regulation Of G Protein-coupled Receptor Signaling Pathway
Regulation Of Systemic Arterial Blood Pressure By Norepinephrine-epinephrine
Positive Regulation Of Mini Excitatory Postsynaptic Potential
Identical Protein Binding
Angiotensin Type I Receptor Activity
Tagcloud
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Tagcloud (Difference)
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Tagcloud (Intersection)
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