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SERPINB8 and PRSS1
Number of citations of the paper that reports this interaction (PubMedID
9402754
)
0
Data Source:
BioGRID
(pull down)
HPRD
(in vitro)
SERPINB8
PRSS1
Description
serpin family B member 8
serine protease 1
Image
No pdb structure
GO Annotations
Cellular Component
Extracellular Space
Cytoplasm
Cytosol
Extracellular Matrix
Extracellular Exosome
Extracellular Region
Extracellular Space
Extracellular Matrix
Blood Microparticle
Molecular Function
Serine-type Endopeptidase Inhibitor Activity
Protein Binding
Peptidase Inhibitor Activity
Serine-type Endopeptidase Activity
Peptidase Activity
Serine-type Peptidase Activity
Hydrolase Activity
Metal Ion Binding
Biological Process
Negative Regulation Of Endopeptidase Activity
Epithelial Cell-cell Adhesion
Proteolysis
Digestion
Extracellular Matrix Disassembly
Pathways
Dissolution of Fibrin Clot
Activation of Matrix Metalloproteinases
Uptake of dietary cobalamins into enterocytes
Developmental Lineage of Pancreatic Acinar Cells
Drugs
2H-Benzimidazol-2-amine
Bis(5-Amidino-Benzimidazolyl)Methane
2-{2-hydroxy-[1,1'-biphenyl]-3-yl}-1H-1,3-benzodiazole-5-carboximidamide
Nalpha-(2-Naphthylsulfonylglycyl)-3-Amidino-D,L-Phenylalanine-Isopropylester
CRA_17693
N-Alpha-(2-Naphthylsulfonyl)-N(3-Amidino-L-Phenylalaninyl)Isopipecolinic Acid Methyl Ester
Hemi-Babim
CRA_10991
Monoisopropylphosphorylserine
[4-(6-Chloro-Naphthalene-2-Sulfonyl)-Piperazin-1-Yl]-(3,4,5,6-Tetrahydro-2h-[1,4']Bipyridinyl-4-Yl)-Methanone
Bis(5-Amidino-2-Benzimidazolyl)Methanone
2-(2-Hydroxy-5-Methoxy-Phenyl)-1h-Benzoimidazole-5-Carboxamidine
5-Amidino-Benzimidazole
Amylamine
CRA_16847
Bis-Benzamidine
CRA_17312
Zk-806450
[4-({[5-Benzyloxy-1-(3-Carbamimidoyl-Benzyl)-1h-Indole-2-Carbonyl]-Amino}-Methyl)-Phenyl]-Trimethyl-Ammonium
2-(2-hydroxy-phenyl)-3H-benzoimidazole-5-carboxamidine
CRA-9334
4-{[1-Methyl-5-(2-Methyl-Benzoimidazol-1-Ylmethyl)-1h-Benzoimidazol-2-Ylmethyl]-Amino}-Benzamidine
CRA_10762
Aminomethylcyclohexane
2-(2-Hydroxy-Phenyl)-1h-Indole-5-Carboxamidine
Benzylamine
CRA_10655
(1R,2S)-2-Phenylcyclopropanaminium
RPR131247
RWJ-56423
CRA_1802
CRA_10972
CRA_1801
[N-[N-(4-Methoxy-2,3,6-trimethylphenylsulfonyl)-L-aspartyl]-D-(4-amidino-phenylalanyl)]-piperidine
Benzamidine
4-Iodobenzo[B]Thiophene-2-Carboxamidine
CRA_8696
CRA_10433
Bis(5-Amidino-2-Benzimidazolyl)Methane Ketone
4-Fluorobenzylamine
RWJ-51084
1-(2-Amidinophenyl)-3-(Phenoxyphenyl)Urea
ZK-806711
3,5-Diiodotyrosine
(2S,3R)-2-[[4-(Tert-butylcarbamoyl)piperazine-1-carbonyl]amino]-6-(diaminomethylideneamino)-3-formylhexanoic acid
bis(5-amidino-benzimidazolyl)methanone zinc
CRA_11092
CRA_9785
Diminazene
CRA_1144
6-Chloro-2-(2-Hydroxy-Biphenyl-3-Yl)-1h-Indole-5-Carboxamidine
Thieno[2,3-B]Pyridine-2-Carboxamidine
Phosphorylisopropane
Zinc;[amino-[2-[[5-[amino(azaniumylidene)methyl]benzimidazol-1-id-2-yl]methyl]benzimidazol-1-id-5-yl]methylidene]azanium
[(1-{2[(4-Carbamimidoyl-Phenylamino)-Methyl]-1-Methyl-1h-Benzoimidazol-5-Yl}-Cyclopropyl)-Pyridin-2-Yl-Methyleneaminooxy]-Acetic Acid Ethyl Ester
N-Alpha-(2-Naphthylsulfonyl)-N(3-Amidino-L-Phenylalaninyl)-4-Acetyl-Piperazine
CRA_9076
N-Alpha-(2-Naphthylsulfonyl)-N-(3-Amidino-L-Phenylalaninyl)-D-Pipecolinic Acid
CRA_23653
Cyclotheonamide A
Bis(5-Amidino-2-Benzimidazolyl)Methane Ketone Hydrate
4-Phenylbutylamine
Phenethylamine
1-(4-Amidinophenyl)-3-(4-Chlorophenyl)Urea
Aeruginosin 98-B
3-Phenylpropylamine
RPR128515
ZK-805623
Imino[2-(2-oxo-1,2-dihydro-3-pyridinyl)-1H-benzimidazol-5-yl]methanaminium
Benzo[B]Thiophene-2-Carboxamidine
CRA_10656
CRA_9678
4-PIPERIDIN-4-YLBUTANAL
2,5-bis-O-{3-[amino(imino)methyl]phenyl}-1,4:3,6-dianhydro-D-glucitol
2-O-(4'-AMIDINOPHENYL)-5-O-(3''-AMIDINOPHENYL)-1,4:3,6-DIANHYDRO-D-SORBITOL
2,5-O,O-BIS-{4',4''-AMIDINOPHENYL}-1,4:3,6-DIANHYDRO-D-SORBITOL
1,4:3,6-Dianhydro-2-O-(3-carbamimidoylphenyl)-5-O-(4-carbamimidoylphenyl)-D-glucitol
Aprotinin
diethyl [(1R)-1,5-diaminopentyl]boronate
(S)-N-(4-carbamimidoylbenzyl)-1-(2-(cyclopentylamino)ethanoyl)pyrrolidine-2-carboxamide
(S)-N-(4-carbamimidoylbenzyl)-1-(2-(cyclohexylamino)ethanoyl)pyrrolidine-2-carboxamide
N-cycloheptylglycyl-N-(4-carbamimidoylbenzyl)-L-prolinamide
6-fluoro-2-(2-hydroxy-3-isobutoxy-phenyl)-1H-benzoimidazole-5-carboxamidine
N-cyclooctylglycyl-N-(4-carbamimidoylbenzyl)-L-prolinamide
2-(2-METHYLPHENYL)-1H-INDOLE-6-CARBOXIMIDAMIDE
2-(3-METHYLPHENYL)-1H-INDOLE-5-CARBOXIMIDAMIDE
(S)-N-(4-carbamimidoylbenzyl)-1-(2-(cyclopentyloxy)ethanoyl)pyrrolidine-2-carboxamide
(S)-N-(4-carbamimidoylbenzyl)-1-(2-(cyclohexyloxy)ethanoyl)pyrrolidine-2-carboxamide
(S)-N-(4-carbamimidoylbenzyl)-1-(3-cyclopentylpropanoyl)pyrrolidine-2-carboxamide
(S)-N-(4-carbamimidoylbenzyl)-1-(3-cyclohexylpropanoyl)pyrrolidine-2-carboxamide
3-{5-[AMINO(IMINIO)METHYL]-1H-INDOL-2-YL}-5-METHOXY-1,1'-BIPHENYL-2-OLATE
4-(METHYLSULFONYL)BENZENECARBOXIMIDAMIDE
5-amino-2,4,6-tribromobenzene-1,3-dicarboxylic acid
+/-METHYL 4-(AMINOIMINOMETHYL)-BETA-[3- INH (AMINOIMINO)PHENYL]BENZENE PENTANOATE
2-(2-METHYLPHENYL)-1H-INDOLE-5-CARBOXIMIDAMIDE
2-Naphthalenesulfonic acid
1-{[1-(2-AMINO-3-PHENYL-PROPIONYL)-PYRROLIDINE-2-CARBONYL]-AMINO}-2-(3-CYANO-PHENYL)-ETHANEBORONIC ACID
[N-(BENZYLOXYCARBONYL)AMINO](4-AMIDINOPHENYL)METHANE-PHOSPHONATE
Nafamostat
Camostat
Diseases
Hereditary pancreatitis; Hereditary chronic pancreatitis
GWAS
Airflow obstruction (
22837378
)
Alcoholic chronic pancreatitis (
28754779
)
Cancer (
29299148
)
Meconium ileus in cystic fibrosis (
30807572
)
Methadone dose in opioid dependence (
28115739
)
Pancreatitis (
23143602
)
Interacting Genes
5 interacting genes:
CAP1
F10
F2
FURIN
PRSS1
11 interacting genes:
DEFA5
LINC00839
PTPN4
RNF26
SERPINA1
SERPINB13
SERPINB8
SERPINF2
SPINK5
TST
UBE3A
Entrez ID
5271
5644
HPRD ID
03412
02039
Ensembl ID
ENSG00000166401
ENSG00000204983
Uniprot IDs
A0A1B0GU38
P50452
P07477
PDB IDs
1FXY
1TRN
2RA3
4WWY
4WXV
7QE8
7QE9
8H3S
Enriched GO Terms of Interacting Partners
?
Serine-type Peptidase Activity
Serine-type Endopeptidase Activity
Golgi Lumen
Peptidase Activity
Extracellular Region
Extracellular Matrix Disassembly
Proteolysis
Endopeptidase Activity
Extracellular Space
Negative Regulation Of Nerve Growth Factor Production
Dibasic Protein Processing
Zymogen Inhibition
Hydrolase Activity
Coagulation
Blood Coagulation
Hemostasis
Blood Microparticle
Golgi Apparatus Subcompartment
Regulation Of Nerve Growth Factor Production
Negative Regulation Of Low-density Lipoprotein Particle Receptor Catabolic Process
Nerve Growth Factor Production
Negative Regulation Of Neurotrophin Production
Negative Regulation Of Proteolysis
Heparin Binding
Negative Regulation Of Receptor Catabolic Process
Thrombospondin Receptor Activity
Viral Translation
Viral Life Cycle
CAMP-mediated Signaling
Neutrophil-mediated Killing Of Gram-negative Bacterium
Cytokine Precursor Processing
Nerve Growth Factor Binding
Regulation Of Low-density Lipoprotein Particle Receptor Catabolic Process
Negative Regulation Of Transforming Growth Factor Beta1 Production
Positive Regulation Of Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Extracellular Matrix Organization
Extracellular Structure Organization
Heparan Sulfate Binding
Regulation Of Body Fluid Levels
Signal Peptide Processing
Endoplasmic Reticulum Lumen
Thrombin-activated Receptor Signaling Pathway
Neutrophil-mediated Killing Of Bacterium
Cytolysis By Host Of Symbiont Cells
Negative Regulation Of Fibrinolysis
Negative Regulation Of Transforming Growth Factor Beta Production
Adenylate Cyclase Binding
Modification Of Postsynaptic Actin Cytoskeleton
Protein Metabolic Process
Negative Regulation Of Cytokine Production
Serine-type Endopeptidase Inhibitor Activity
Peptidase Inhibitor Activity
Negative Regulation Of Proteolysis
Regulation Of Proteolysis
Negative Regulation Of Endopeptidase Activity
Protease Binding
Negative Regulation Of Peptidase Activity
Regulation Of Endopeptidase Activity
Extracellular Space
Acute-phase Response
Negative Regulation Of Hydrolase Activity
Negative Regulation Of Protein Metabolic Process
Negative Regulation Of Keratinocyte Apoptotic Process
Endopeptidase Inhibitor Activity
Sperm Entry
Positive Regulation Of Golgi Lumen Acidification
Negative Regulation Of Antibacterial Peptide Production
Acute Inflammatory Response
Platelet Alpha Granule Lumen
Cyanate Catabolic Process
3-mercaptopyruvate Sulfurtransferase Activity
RRNA Transport
Thiosulfate-cyanide Sulfurtransferase Activity
RRNA Import Into Mitochondrion
Regulation Of Golgi Lumen Acidification
Tagcloud
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Tagcloud (Intersection)
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