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GRK5 and AVPR1A
Number of citations of the paper that reports this interaction (PubMedID
10858434
)
0
Data Source:
HPRD
(in vitro, in vivo)
GRK5
AVPR1A
Description
G protein-coupled receptor kinase 5
arginine vasopressin receptor 1A
Image
GO Annotations
Cellular Component
Nucleus
Cytoplasm
Cytosol
Plasma Membrane
Membrane
Nuclear Speck
Nuclear Membrane
Endosome
Plasma Membrane
Membrane
Endocytic Vesicle
Molecular Function
Nucleotide Binding
Protein Kinase Activity
Protein Serine/threonine Kinase Activity
G Protein-coupled Receptor Kinase Activity
Protein Kinase C Binding
Protein Binding
ATP Binding
Phospholipid Binding
Lipid Binding
Kinase Activity
Transferase Activity
Beta-adrenergic Receptor Kinase Activity
G Protein-coupled Receptor Activity
Vasopressin Receptor Activity
Protein Kinase C Binding
Protein Binding
G Protein-coupled Peptide Receptor Activity
Peptide Hormone Binding
V1A Vasopressin Receptor Binding
Biological Process
Apoptotic Process
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
Tachykinin Receptor Signaling Pathway
Regulation Of G Protein-coupled Receptor Signaling Pathway
Positive Regulation Of Cell Population Proliferation
Regulation Of Signal Transduction
Wnt Signaling Pathway
Negative Regulation Of Apoptotic Process
Fat Cell Differentiation
Protein Autophosphorylation
Regulation Of Cell Cycle
Regulation Of Systemic Arterial Blood Pressure By Vasopressin
Maternal Aggressive Behavior
Positive Regulation Of Systemic Arterial Blood Pressure
Generation Of Precursor Metabolites And Energy
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
Positive Regulation Of Cytosolic Calcium Ion Concentration
Negative Regulation Of Female Receptivity
Grooming Behavior
Blood Circulation
Regulation Of Blood Pressure
Positive Regulation Of Cell Population Proliferation
Positive Regulation Of Heart Rate
Positive Regulation Of Glutamate Secretion
Myotube Differentiation
Calcium-mediated Signaling
Telencephalon Development
Positive Regulation Of Cell Growth
Positive Regulation Of Prostaglandin Biosynthetic Process
Positive Regulation Of Cellular PH Reduction
Cellular Response To Hormone Stimulus
Social Behavior
Cellular Response To Water Deprivation
Maternal Behavior
Sperm Ejaculation
Positive Regulation Of Blood Pressure
Positive Regulation Of Vasoconstriction
Response To Corticosterone
Negative Regulation Of Transmission Of Nerve Impulse
Transport Across Blood-brain Barrier
Pathways
G alpha (q) signalling events
G alpha (s) signalling events
Vasopressin-like receptors
G alpha (q) signalling events
Defective AVP does not bind AVPR1A,B and causes neurohypophyseal diabetes insipidus (NDI)
Drugs
Desmopressin
Vasopressin
Felypressin
Conivaptan
Terlipressin
PH-284
Tolvaptan
Atosiban
Relcovaptan
Lypressin
Pecavaptan
Diseases
GWAS
Appendicular lean mass (
33097823
)
Coronary artery aneurysm in Kawasaki disease (
27171184
)
Early onset periodontitis x smoking status interaction (
31537151
)
Height (
28552196
)
Lymphocyte count (
32888494
)
Lymphocyte percentage of white cells (
32888494
)
Mean platelet volume (
27863252
32888494
)
Methadone dose in opioid dependence (
30060048
)
Neutrophil percentage of white cells (
32888494
)
Obesity-related traits (
23251661
)
Platelet count (
32888494
)
Platelet distribution width (
27863252
32888494
)
Risky sexual behaviors in alcohol dependence (
28990359
)
Thrombin-induced platelet aggregation (
32649856
)
Thymus and reactivation regulated chemokine levels (
33227023
)
Type 2 diabetes (
22961080
)
Venous thromboembolism (
31676865
31420334
)
Waist circumference adjusted for body mass index (
34021172
)
Chronotype (
30696823
)
Diastolic blood pressure x smoking status (ever vs never) interaction (2df test) (
29455858
)
Hippocampal volume (
29860282
)
Morning person (
30696823
)
Type 2 diabetes (
31049640
)
Interacting Genes
19 interacting genes:
ADRB2
AGTR1
AVPR1A
AVPR1B
AVPR2
BDKRB2
CABP1
CALM1
CAV1
CHRM2
DLGAP2
GIT1
RCVRN
RHO
SNCA
SNCB
SNCG
TACR1
TBXA2R
3 interacting genes:
AVP
GRK5
PRKCA
Entrez ID
2869
552
HPRD ID
02926
02894
Ensembl ID
ENSG00000198873
ENSG00000166148
Uniprot IDs
P34947
P37288
X5D2B0
PDB IDs
4TNB
4TND
6PJX
8UAP
8UAQ
9BRE
9BRG
9BRH
9BRI
9BRJ
1YTV
Enriched GO Terms of Interacting Partners
?
Regulation Of Vasoconstriction
Blood Vessel Diameter Maintenance
Regulation Of Tube Size
Regulation Of Blood Circulation
Positive Regulation Of Vasoconstriction
G Protein-coupled Receptor Activity
Regulation Of System Process
G Protein-coupled Receptor Signaling Pathway
Vascular Process In Circulatory System
Circulatory System Process
Regulation Of Systemic Arterial Blood Pressure Mediated By A Chemical Signal
Positive Regulation Of Cytosolic Calcium Ion Concentration
System Process
Regulation Of Blood Pressure
Regulation Of Systemic Arterial Blood Pressure
Regulation Of Smooth Muscle Contraction
Regulation Of Transport
Regulation Of Systemic Arterial Blood Pressure By Vasopressin
Regulation Of Muscle Contraction
Modulation Of Chemical Synaptic Transmission
Positive Regulation Of Blood Pressure
Vasopressin Receptor Activity
Regulation Of Cell Communication
Cuprous Ion Binding
Presynaptic Endocytosis
Regulation Of Muscle System Process
Smooth Muscle Contraction
Regulation Of Signaling
Regulation Of Small Molecule Metabolic Process
Regulation Of Multicellular Organismal Process
Regulation Of Biological Quality
Plasma Membrane
Regulation Of Secretion
Vesicle-mediated Transport In Synapse
Endocytosis
Sperm Ejaculation
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Endosome
Synaptic Vesicle Endocytosis
Signal Transduction
Membrane
Chemical Synaptic Transmission
Sperm Midpiece
Positive Regulation Of Small Molecule Metabolic Process
Regulation Of Secretion By Cell
Trans-synaptic Signaling
Regulation Of Metal Ion Transport
Synaptic Signaling
Axon Terminus
Aggressive Behavior
Renal Absorption
Protein Kinase Activity
Response To Ethanol
Positive Regulation Of Cell Population Proliferation
Negative Regulation Of Programmed Cell Death
Negative Regulation Of Apoptotic Process
Renal System Process
V1B Vasopressin Receptor Binding
Regulation Of G Protein-coupled Receptor Signaling Pathway
V1A Vasopressin Receptor Binding
Regulation Of Programmed Cell Death
Regulation Of Apoptotic Process
Adenylate Cyclase-modulating G Protein-coupled Receptor Signaling Pathway
Negative Regulation Of Female Receptivity
Neurohypophyseal Hormone Activity
Response To Ketone
Response To Alcohol
Maternal Aggressive Behavior
Beta-adrenergic Receptor Kinase Activity
Calcium,diacylglycerol-dependent Serine/threonine Kinase Activity
Positive Regulation Of Dense Core Granule Biogenesis
Positive Regulation Of Angiotensin-activated Signaling Pathway
Histone H3T6 Kinase Activity
Alphav-beta3 Integrin-PKCalpha Complex
Protein Kinase C Signaling
Positive Regulation Of Cellular PH Reduction
Regulation Of Cell Population Proliferation
Positive Regulation Of Secretion By Cell
Regulation Of Angiotensin-activated Signaling Pathway
Positive Regulation Of Secretion
Renal Water Absorption
Negative Regulation Of Transmission Of Nerve Impulse
Positive Regulation Of Adenylate Cyclase-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of Female Receptivity
Renal Water Transport
Female Mating Behavior
Aggressive Behavior
Response To 2,3,7,8-tetrachlorodibenzodioxine
Tachykinin Receptor Signaling Pathway
Protein Phosphorylation
G Protein-coupled Receptor Kinase Activity
Desmosome Assembly
Phosphorylation
Signaling Receptor Binding
Positive Regulation Of Prostaglandin Biosynthetic Process
Protein Serine/threonine Kinase Activity
Negative Regulation Of Glial Cell Apoptotic Process
Positive Regulation Of Unsaturated Fatty Acid Biosynthetic Process
Positive Regulation Of Glutamate Secretion
Mitotic Nuclear Membrane Disassembly
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Tagcloud (Difference)
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Tagcloud (Intersection)
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