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SRC and AHR
Number of citations of the paper that reports this interaction (PubMedID
10947077
)
65
Data Source:
BioGRID
(pull down)
SRC
AHR
Description
SRC proto-oncogene, non-receptor tyrosine kinase
aryl hydrocarbon receptor
Image
GO Annotations
Cellular Component
Podosome
Nucleus
Cytoplasm
Mitochondrion
Mitochondrial Inner Membrane
Lysosome
Late Endosome
Cytosol
Cytoskeleton
Actin Filament
Plasma Membrane
Caveola
Cell-cell Junction
Focal Adhesion
Membrane
Cell Junction
Ruffle Membrane
Membrane Raft
Perinuclear Region Of Cytoplasm
Extracellular Exosome
Anchoring Junction
Chromatin
Nucleus
Nucleoplasm
Transcription Regulator Complex
Cytoplasm
Cytosol
Protein-containing Complex
Aryl Hydrocarbon Receptor Complex
Cytosolic Aryl Hydrocarbon Receptor Complex
Nuclear Aryl Hydrocarbon Receptor Complex
Molecular Function
Nucleotide Binding
Protein Kinase Activity
Protein Tyrosine Kinase Activity
Non-membrane Spanning Protein Tyrosine Kinase Activity
Signaling Receptor Binding
Integrin Binding
Protein Binding
ATP Binding
Phospholipase Activator Activity
Kinase Activity
Transferase Activity
Enzyme Binding
Protein Domain Specific Binding
Heme Binding
Protein Tyrosine Kinase Activator Activity
Signaling Receptor Activator Activity
Ionotropic Glutamate Receptor Binding
SH2 Domain Binding
Phospholipase Binding
Transmembrane Transporter Binding
Cadherin Binding
Ephrin Receptor Binding
ATPase Binding
Phosphoprotein Binding
BMP Receptor Binding
Connexin Binding
Scaffold Protein Binding
Transcription Cis-regulatory Region Binding
DNA-binding Transcription Factor Activity, RNA Polymerase II-specific
Cis-regulatory Region Sequence-specific DNA Binding
TFIID-class Transcription Factor Complex Binding
Transcription Coactivator Binding
DNA Binding
DNA-binding Transcription Factor Activity
Nuclear Receptor Activity
Protein Binding
TBP-class Protein Binding
Protein Homodimerization Activity
Protein Heterodimerization Activity
Protein Dimerization Activity
Hsp90 Protein Binding
RNA Polymerase II-specific DNA-binding Transcription Factor Binding
E-box Binding
Sequence-specific Double-stranded DNA Binding
Biological Process
Negative Regulation Of Transcription By RNA Polymerase II
Stimulatory C-type Lectin Receptor Signaling Pathway
Neutrophil Activation Involved In Immune Response
Immune System Process
Negative Regulation Of Inflammatory Response To Antigenic Stimulus
Cell Adhesion
Signal Transduction
Signal Complex Assembly
Epidermal Growth Factor Receptor Signaling Pathway
Transforming Growth Factor Beta Receptor Signaling Pathway
Integrin-mediated Signaling Pathway
Regulation Of Epithelial Cell Migration
Positive Regulation Of Epithelial Cell Migration
Positive Regulation Of Protein Processing
Macroautophagy
Cell Migration
Protein Deubiquitination
Peptidyl-tyrosine Phosphorylation
Regulation Of Cell-cell Adhesion
Cell Differentiation
Platelet Activation
Forebrain Development
T Cell Costimulation
Negative Regulation Of Protein-containing Complex Assembly
Protein Destabilization
Cellular Response To Nutrient Levels
Negative Regulation Of Telomere Maintenance
Regulation Of Intracellular Estrogen Receptor Signaling Pathway
Positive Regulation Of Integrin Activation
Toll-like Receptor 3 Signaling Pathway
Regulation Of Toll-like Receptor 3 Signaling Pathway
Substrate Adhesion-dependent Cell Spreading
Cellular Response To Reactive Oxygen Species
Positive Regulation Of Dephosphorylation
Negative Regulation Of Hippo Signaling
Intracellular Signal Transduction
Osteoclast Development
Cellular Response To Platelet-derived Growth Factor Stimulus
Fc-gamma Receptor Signaling Pathway Involved In Phagocytosis
ERBB2 Signaling Pathway
Angiotensin-activated Signaling Pathway
TORC1 Signaling
Vasodilation
Odontogenesis
Negative Regulation Of Apoptotic Process
Regulation Of Vascular Permeability
Stress Fiber Assembly
Proteasome-mediated Ubiquitin-dependent Protein Catabolic Process
Regulation Of Bone Resorption
Bone Resorption
Positive Regulation Of Notch Signaling Pathway
Positive Regulation Of Glycolytic Process
Symbiont Entry Into Host Cell
Protein Autophosphorylation
Vascular Endothelial Growth Factor Receptor Signaling Pathway
Ephrin Receptor Signaling Pathway
Focal Adhesion Assembly
Oogenesis
Progesterone Receptor Signaling Pathway
Leukocyte Migration
Positive Regulation Of Small GTPase Mediated Signal Transduction
Negative Regulation Of Focal Adhesion Assembly
Positive Regulation Of Phosphatidylinositol 3-kinase/protein Kinase B Signal Transduction
Negative Regulation Of Mitochondrial Depolarization
Uterus Development
Branching Involved In Mammary Gland Duct Morphogenesis
Regulation Of Cell Projection Assembly
Intestinal Epithelial Cell Development
Interleukin-6-mediated Signaling Pathway
Cellular Response To Hydrogen Peroxide
Positive Regulation Of ERK1 And ERK2 Cascade
Response To Interleukin-1
Cellular Response To Peptide Hormone Stimulus
Cellular Response To Progesterone Stimulus
Cellular Response To Fluid Shear Stress
Cellular Response To Transforming Growth Factor Beta Stimulus
Positive Regulation Of Podosome Assembly
Positive Regulation Of Protein Serine/threonine Kinase Activity
Regulation Of Heart Rate By Cardiac Conduction
Positive Regulation Of Canonical Wnt Signaling Pathway
Positive Regulation Of Protein Localization To Nucleus
Negative Regulation Of Neutrophil Activation
Negative Regulation Of TORC1 Signaling
Positive Regulation Of TORC1 Signaling
Positive Regulation Of Lamellipodium Morphogenesis
Positive Regulation Of Platelet-derived Growth Factor Receptor-beta Signaling Pathway
Regulation Of Early Endosome To Late Endosome Transport
Negative Regulation Of Anoikis
Negative Regulation Of Extrinsic Apoptotic Signaling Pathway
Negative Regulation Of Intrinsic Apoptotic Signaling Pathway
Regulation Of Caveolin-mediated Endocytosis
Blood Vessel Development
Regulation Of Adaptive Immune Response
Negative Regulation Of T Cell Mediated Immune Response To Tumor Cell
Regulation Of DNA-templated Transcription
Regulation Of Transcription By RNA Polymerase II
Xenobiotic Metabolic Process
Apoptotic Process
Response To Xenobiotic Stimulus
Response To Toxic Substance
Regulation Of Gene Expression
Intracellular Receptor Signaling Pathway
Regulation Of B Cell Proliferation
Circadian Regulation Of Gene Expression
Negative Regulation Of DNA-templated Transcription
Positive Regulation Of DNA-templated Transcription
Positive Regulation Of Transcription By RNA Polymerase II
Rhythmic Process
Negative Regulation Of Inflammatory Response
Intestinal Epithelial Structure Maintenance
Cellular Response To Molecule Of Bacterial Origin
Cellular Response To CAMP
Cellular Response To Forskolin
Cellular Response To 2,3,7,8-tetrachlorodibenzodioxine
Pathways
Signaling by ERBB2
Nuclear signaling by ERBB4
Downregulation of ERBB4 signaling
PIP3 activates AKT signaling
GAB1 signalosome
Downstream signal transduction
Constitutive Signaling by Aberrant PI3K in Cancer
Integrin signaling
GRB2:SOS provides linkage to MAPK signaling for Integrins
p130Cas linkage to MAPK signaling for integrins
G alpha (s) signalling events
G alpha (i) signalling events
G alpha (i) signalling events
DCC mediated attractive signaling
DCC mediated attractive signaling
Netrin mediated repulsion signals
Regulation of commissural axon pathfinding by SLIT and ROBO
RAF activation
MAP2K and MAPK activation
Signaling by moderate kinase activity BRAF mutants
Signaling by high-kinase activity BRAF mutants
Signaling by BRAF and RAF1 fusions
Paradoxical activation of RAF signaling by kinase inactive BRAF
PI5P, PP2A and IER3 Regulate PI3K/AKT Signaling
MET activates PTK2 signaling
InlA-mediated entry of Listeria monocytogenes into host cells
Regulation of RUNX1 Expression and Activity
RUNX2 regulates osteoblast differentiation
Regulation of RUNX3 expression and activity
Extra-nuclear estrogen signaling
RHOU GTPase cycle
Activated NTRK2 signals through FYN
Activated NTRK3 signals through PI3K
Activated NTRK3 signals through PI3K
Long-term potentiation
GPER1 signaling
Signaling downstream of RAS mutants
Signaling by RAF1 mutants
Signaling by CSF1 (M-CSF) in myeloid cells
Degradation of CDH1
PPARA activates gene expression
Phase I - Functionalization of compounds
Endogenous sterols
Xenobiotics
Aryl hydrocarbon receptor signalling
Drugs
Dasatinib
RU84687
RU79256
N6-Benzyl Adenosine-5'-Diphosphate
RU85493
RU78262
Phosphonotyrosine
Malonic acid
RU83876
RU90395
RU79072
RU78783
1-Tert-Butyl-3-(4-Chloro-Phenyl)-1h-Pyrazolo[3,4-D]Pyrimidin-4-Ylamine
PASBN
2-[4-[(Z)-2-Acetamido-3-oxo-3-[[(3S)-2-oxo-1-[(4-phenylphenyl)methyl]azepan-3-yl]amino]prop-1-enyl]-2-formylphenyl]acetic acid
PAS219
DPI59
RU82197
Phenylphosphate
RU78300
RU79073
RU82209
ISO24
RU85053
RU78299
Oxalic Acid
RU78191
Citric acid
Paratoulene phosphate
4-[(4-METHYL-1-PIPERAZINYL)METHYL]-N-[3-[[4-(3-PYRIDINYL)-2-PYRIMIDINYL]AMINO]PHENYL]-BENZAMIDE
Purvalanol A
XL228
Tirbanibulin
Bosutinib
1-[1-(3-aminophenyl)-3-tert-butyl-1H-pyrazol-5-yl]-3-naphthalen-1-ylurea
1-[1-(3-aminophenyl)-3-tert-butyl-1H-pyrazol-5-yl]-3-phenylurea
3-[4-AMINO-1-(1-METHYLETHYL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-3-YL]PHENOL
PD-168393
[4-({4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile
PP-121
1-cyclobutyl-3-(3,4-dimethoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(1-methylethyl)-3-quinolin-6-yl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-CARCOXY-5-ISOPROPYLTHIAZOLYL)BENZOPIPERIDINE
N-(4-PHENYLAMINO-QUINAZOLIN-6-YL)-ACRYLAMIDE
(2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide
Ponatinib
Nintedanib
Fostamatinib
Omeprazole
Mexiletine
Nimodipine
Flutamide
Atorvastatin
Leflunomide
Ginseng
Indirubin-3'-monoxime
Resveratrol
Quercetin
Tapinarof
beta-Naphthoflavone
Emodin
1-[(4S)-4-amino-5-(1,3-benzothiazol-2-yl)-5-oxopentyl]guanidine
Diosmin
Kynurenic Acid
Epigallocatechin gallate
Cantharidin
Indirubin
Carbendazim
Indigo
Diseases
GWAS
L1-L4 bone mineral density x serum urate levels interaction (
34046847
)
Retinopathy in non-diabetics (
23393555
)
Rheumatoid arthritis (
30891314
)
Squamous cell carcinoma (
26908436
)
Alanine aminotransferase (ALT) levels after remission induction therapy in actute lymphoblastic leukemia (ALL) (
28090653
)
Bitter beverage consumption (
31046077
)
Bitter non-alcoholic beverage consumption (
31046077
)
Caffeine consumption (
21490707
)
Caffeine consumption from coffee (
33287642
)
Caffeine consumption from coffee or tea (
33287642
)
Caffeine consumption from tea (
33287642
)
Caffeine metabolism (plasma 1,3,7-trimethylxanthine (caffeine) level) (
27702941
)
Caffeine metabolism (plasma 1,7-dimethylxanthine (paraxanthine) to 1,3,7-trimethylxanthine (caffeine) ratio) (
27702941
)
Coffee consumption (
31046077
25288136
21357676
29367735
31345160
31959922
)
Coffee consumption (cups per day) (
25288136
31837886
)
Cutaneous malignant melanoma (
32341527
)
Cutaneous squamous cell carcinoma (
32041948
27424798
)
Estimated glomerular filtration rate (
31152163
)
HDL cholesterol levels (
32203549
)
Inflammatory bowel disease (
26192919
)
Lung cancer in ever smokers (
28604730
)
Metabolic traits (
21886157
)
Microalbuminuria (
31511532
)
Plasma kynurenine levels in major depressive disorder (
29317604
)
Rosacea symptom severity (
29771307
)
Severe influenza A (H1N1) infection (
26379185
)
Sweet beverage consumption (
31046077
)
Tea consumption (
31046077
)
Triglyceride levels (
32203549
)
Ulcerative colitis (
26192919
)
Urinary albumin excretion (
30220432
)
Urinary albumin excretion (no hypertensive medication) (
30220432
)
Urinary albumin-to-creatinine ratio (
30910378
31630189
31511532
)
Urinary potassium excretion (
31409800
)
Urinary sodium excretion (
31409800
)
Interacting Genes
303 interacting genes:
ABL1
ACTN1
ADAM12
ADAM15
ADRB2
ADRB3
AFAP1
AFAP1L2
AGAP1
AHR
AKT1
ALDOB
ANKRD11
ANXA1
ANXA2
ANXA7
AR
ARHGAP1
ARHGAP17
ARHGAP32
ARHGAP35
ARR3
ASAP1
ATG9A
ATP2B4
AXL
BAAT
BCAR1
BCCIP
BCR
BMX
BRMS1
CA3
CASP8
CAV1
CAV2
CBL
CBLC
CCDC180
CCNA1
CD2AP
CD33
CD36
CD44
CD46
CD47
CD59
CDC25A
CDCP1
CDH5
CDK1
CDK5
CDKN1B
CEACAM1
CEACAM3
CFL1
CHUK
CLTC
CNTNAP1
COASY
CORO7
CRMP1
CSK
CTNNB1
CTNND1
CTSV
CTTN
DAB1
DAB2
DAG1
DAPP1
DDR2
DGKA
DGKZ
DLG4
DNM1
DNM2
DOK1
DOK2
DOK4
DUSP12
EFNA5
EFNB1
EFNB2
EFS
EGFR
EGLN1
EMD
ENO1
EPHA3
EPHA4
EPHB2
EPS8
ERBB2
ERBB3
ERBB4
ERRFI1
ESR1
ESR2
ETS1
ETS2
EVL
FANCC
FARP2
FASLG
FBP2
FBXO5
FGR
FHIT
FLNA
FLT3
FOXO1
FRS2
FYB1
FZR1
GAB1
GAB2
GAB3
GALNT12
GFAP
GIT1
GJA1
GJB1
GRB10
GRB2
GRIN2A
GRIN2B
GRK2
GTF2I
GUCY2C
HDAC3
HEMGN
HLA-A
HLA-B
HNF1A
HNRNPK
HRAS
HSP90AA1
IGF1R
IKBKB
IKBKG
IL6R
INPPL1
INSR
ITGB3
ITK
JUP
KCNA5
KCNB1
KCNQ5
KDR
KHDRBS1
KIFAP3
KIT
LATS2
LRP1
MAP2
MAP2K1
MAPK15
MAPK3
MAPK8IP3
MAPRE1
MAPT
MATK
MDM2
MED28
MET
MICAL1
MPZL1
MST1R
MT-ND2
MUC1
MYLK
NANS
NCOA6
NEDD4
NFKBIA
NMT1
NOS2
NPHS1
NR1I2
NR1I3
NR3C1
P2RY2
PAK2
PDCD6IP
PDE4D
PDE6G
PDGFRB
PDPK1
PECAM1
PELP1
PGR
PIK3R1
PIK3R3
PIP5K1C
PKD1
PLCG1
PLD1
PLD2
PLSCR1
PPARD
PPARGC1B
PPP2CB
PRKACA
PRKCA
PRKCD
PRKCE
PRKCH
PRKCI
PRKCZ
PRKD1
PROM1
PTK2
PTK2B
PTPA
PTPN1
PTPN11
PTPN18
PTPN2
PTPN21
PTPN6
PTPRA
PTPRC
PTPRE
PXN
RACK1
RAF1
RARA
RASA1
RASGRF1
RET
RGS16
RPL10
RPS6KA3
RPS6KB1
RPS6KB2
RXRA
SH2D3C
SH3BP1
SH3PXD2A
SHB
SHC1
SKAP1
SKAP2
SLC9A2
SMARCB1
SMARCE1
SNCA
SOCS1
SORBS1
SPTAN1
SRCIN1
SRF
SRPK2
STAP2
STAT1
STAT3
STAT5A
STAT5B
STAT6
STUB1
STX17
SYK
SYN1
TAMALIN
TERT
THRA
THRB
TIAM1
TMPO
TNFRSF11A
TNFRSF1A
TNK2
TP53
TRAF1
TRAF3
TRAF6
TRAT1
TRIM50
TRIM7
TRIP10
TRIP6
TRPC6
TRPV4
TUB
TXK
TYRO3
USP8
VCL
VDR
VIL1
WAS
WASL
WBP11
WWOX
XPA
YTHDC1
YWHAB
YWHAE
YWHAG
YWHAH
ZNF189
35 interacting genes:
AIP
AR
ARNT
ARNT2
BMAL1
CCNT1
CUL4B
DAP3
EP300
ESR1
GTF2F1
GTF2F2
HSP90AA1
IVNS1ABP
NCOA1
NCOA2
NCOA7
NCOR2
NEDD8
NR2F1
NRIP1
PTGES3
RB1
RELA
SMARCA4
SP1
SRC
STUB1
TAF4
TAF6
TAF7
TAF9
TBL3
TBP
XPO1
Entrez ID
6714
196
HPRD ID
01819
02596
Ensembl ID
ENSG00000197122
ENSG00000106546
Uniprot IDs
P12931
P35869
PDB IDs
1A07
1A08
1A09
1A1A
1A1B
1A1C
1A1E
1FMK
1HCS
1HCT
1KSW
1O41
1O42
1O43
1O44
1O45
1O46
1O47
1O48
1O49
1O4A
1O4B
1O4C
1O4D
1O4E
1O4F
1O4G
1O4H
1O4I
1O4J
1O4K
1O4L
1O4M
1O4N
1O4O
1O4P
1O4Q
1O4R
1SHD
1Y57
1YI6
1YOJ
1YOL
1YOM
2BDF
2BDJ
2H8H
2SRC
3VRO
3ZMP
3ZMQ
4F59
4F5A
4F5B
4HXJ
4K11
4MXO
4MXX
4MXY
4MXZ
6ATE
6C4S
6E6E
6EHJ
7NG7
7OTE
7T1U
7YQE
8GWH
8HAQ
8JF3
8JN8
8JN9
8VCF
8VCG
5NJ8
7ZUB
8QMO
Enriched GO Terms of Interacting Partners
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Signal Transduction
Cell Surface Receptor Signaling Pathway
Cell Surface Receptor Protein Tyrosine Kinase Signaling Pathway
Regulation Of Signaling
Plasma Membrane
Regulation Of Cell Communication
Regulation Of Signal Transduction
Enzyme-linked Receptor Protein Signaling Pathway
Regulation Of Multicellular Organismal Process
Regulation Of Intracellular Signal Transduction
Intracellular Signal Transduction
Regulation Of Cellular Component Organization
Regulation Of Programmed Cell Death
Regulation Of Apoptotic Process
Positive Regulation Of Signal Transduction
Positive Regulation Of Intracellular Signal Transduction
Positive Regulation Of Signaling
Cytosol
Cytoplasm
Regulation Of Developmental Process
Positive Regulation Of Cell Communication
Regulation Of Transport
Positive Regulation Of Multicellular Organismal Process
Positive Regulation Of Metabolic Process
Intracellular Signaling Cassette
Developmental Process
Positive Regulation Of Macromolecule Metabolic Process
Focal Adhesion
Protein Kinase Activity
Protein Tyrosine Kinase Activity
Negative Regulation Of Programmed Cell Death
Kinase Activity
Regulation Of Cell Population Proliferation
Regulation Of Locomotion
Negative Regulation Of Signaling
Negative Regulation Of Apoptotic Process
Cellular Response To Oxygen-containing Compound
Negative Regulation Of Cell Communication
Regulation Of MAPK Cascade
Regulation Of Cell Adhesion
Regulation Of Multicellular Organismal Development
Regulation Of Immune System Process
Positive Regulation Of Biosynthetic Process
Regulation Of Cell Motility
Regulation Of Cell Migration
Negative Regulation Of Signal Transduction
Regulation Of Cell Differentiation
Regulation Of Biological Quality
Positive Regulation Of Immune System Process
Phosphorylation
Aryl Hydrocarbon Receptor Binding
Positive Regulation Of Nucleobase-containing Compound Metabolic Process
Nucleoplasm
Positive Regulation Of Transcription By RNA Polymerase II
DNA-templated Transcription
Positive Regulation Of RNA Biosynthetic Process
Positive Regulation Of DNA-templated Transcription
Transcription By RNA Polymerase II
Regulation Of Transcription By RNA Polymerase II
Positive Regulation Of Macromolecule Metabolic Process
Positive Regulation Of Macromolecule Biosynthetic Process
Positive Regulation Of RNA Metabolic Process
Regulation Of Primary Metabolic Process
Positive Regulation Of Biosynthetic Process
Regulation Of Nucleobase-containing Compound Metabolic Process
Positive Regulation Of Metabolic Process
Regulation Of DNA-templated Transcription
Regulation Of RNA Biosynthetic Process
Nucleobase-containing Compound Biosynthetic Process
Regulation Of Macromolecule Metabolic Process
Regulation Of RNA Metabolic Process
Macromolecule Biosynthetic Process
Regulation Of Metabolic Process
Transcription Regulator Complex
RNA Polymerase II General Transcription Initiation Factor Activity
MRNA Transcription By RNA Polymerase II
Regulation Of Macromolecule Biosynthetic Process
Protein-containing Complex
Nucleus
Nucleic Acid Metabolic Process
MRNA Transcription
Regulation Of Gene Expression
Transcription Preinitiation Complex Assembly
Transcription Factor TFIID Complex
DNA-binding Transcription Factor Binding
Chromatin
DNA-templated Transcription Initiation
Nuclear Receptor Binding
RNA Metabolic Process
DNA Binding
Transcription Initiation At RNA Polymerase II Promoter
RNA Polymerase II Preinitiation Complex Assembly
Intracellular Receptor Signaling Pathway
Aryl Hydrocarbon Receptor Complex
Nucleobase-containing Compound Metabolic Process
RNA Polymerase II-specific DNA-binding Transcription Factor Binding
Transcription Coactivator Activity
Regulation Of Protein Metabolic Process
Regulation Of Intracellular Steroid Hormone Receptor Signaling Pathway
Negative Regulation Of Transcription By RNA Polymerase II
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Tagcloud (Intersection)
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