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HTR2A
Description
5-hydroxytryptamine receptor 2A
Image
GO Annotations
Cellular Component
Neurofilament
Plasma Membrane
Caveola
Membrane
Axon
Dendrite
Cytoplasmic Vesicle
Presynaptic Membrane
Cell Projection
Neuronal Cell Body
Dendritic Shaft
Synapse
Postsynaptic Membrane
Cell Body Fiber
G Protein-coupled Serotonin Receptor Complex
Presynapse
Glutamatergic Synapse
Molecular Function
Gq/11-coupled Serotonin Receptor Activity
Virus Receptor Activity
G Protein-coupled Receptor Activity
G Protein-coupled Serotonin Receptor Activity
Protein Binding
Protein Tyrosine Kinase Activator Activity
Neurotransmitter Receptor Activity
Identical Protein Binding
Protein-containing Complex Binding
Serotonin Binding
1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine Binding
Serotonin Receptor Activity
Biological Process
Temperature Homeostasis
Positive Regulation Of Cytokine Production Involved In Immune Response
Glycolytic Process
Intracellular Calcium Ion Homeostasis
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
G Protein-coupled Receptor Signaling Pathway, Coupled To Cyclic Nucleotide Second Messenger
Positive Regulation Of Cytosolic Calcium Ion Concentration
Phospholipase C-activating Serotonin Receptor Signaling Pathway
Serotonin Receptor Signaling Pathway
Chemical Synaptic Transmission
Memory
Positive Regulation Of Cell Population Proliferation
Response To Xenobiotic Stimulus
Positive Regulation Of Phosphatidylinositol Biosynthetic Process
Regulation Of Dopamine Secretion
Artery Smooth Muscle Contraction
Urinary Bladder Smooth Muscle Contraction
Positive Regulation Of Heat Generation
Response To Cocaine
Negative Regulation Of Potassium Ion Transport
Positive Regulation Of Neuron Apoptotic Process
Protein Localization To Cytoskeleton
Positive Regulation Of Fat Cell Differentiation
Positive Regulation Of Glycolytic Process
Positive Regulation Of Vasoconstriction
Symbiont Entry Into Host Cell
Sensitization
Behavioral Response To Cocaine
Positive Regulation Of Inflammatory Response
Sensory Perception Of Temperature Stimulus
Detection Of Temperature Stimulus Involved In Sensory Perception Of Pain
Detection Of Mechanical Stimulus Involved In Sensory Perception Of Pain
Release Of Sequestered Calcium Ion Into Cytosol
Negative Regulation Of Synaptic Transmission, Glutamatergic
Positive Regulation Of ERK1 And ERK2 Cascade
G Protein-coupled Serotonin Receptor Signaling Pathway
Presynaptic Modulation Of Chemical Synaptic Transmission
Positive Regulation Of Execution Phase Of Apoptosis
Positive Regulation Of Platelet Aggregation
Positive Regulation Of DNA Biosynthetic Process
Pathways
Serotonin receptors
G alpha (q) signalling events
Drugs
Ziprasidone
Methysergide
Cabergoline
Zolmitriptan
Dihydroergotamine
Amitriptyline
Olanzapine
Clozapine
Mirtazapine
Loxapine
Remoxipride
Promazine
Cyproheptadine
Imipramine
Chlorpromazine
Chlorpromazine
Haloperidol
Nortriptyline
Amoxapine
Lamotrigine
Fenfluramine
Lisuride
Cisapride
Fluphenazine
Trazodone
Thioridazine
Ergotamine
Apomorphine
Paroxetine
Paroxetine
Trimipramine
Risperidone
Epinastine
Propiomazine
Minaprine
Donepezil
Flupentixol
Cyclobenzaprine
Mesoridazine
Maprotiline
Ergoloid mesylate
Tegaserod
Doxepin
Nefazodone
Desipramine
Escitalopram
Pergolide
Bromocriptine
Ketamine
Quetiapine
Aripiprazole
Chlorprothixene
Chlorprothixene
Clomipramine
Paliperidone
Yohimbine
Methotrimeprazine
MMDA
Midomafetamine
Dimethyltryptamine
4-Bromo-2,5-dimethoxyphenethylamine
Acepromazine
Molindone
Pipotiazine
Thiothixene
Zuclopenthixol
Aniracetam
Fluspirilene
Flibanserin
Iloperidone
HY10275
APD791
Pimavanserin
Epicept NP-1
BL-1020
Cariprazine
Lumateperone
YKP-1358
Sertindole
Mianserin
Pizotifen
Asenapine
Ocaperidone
Amisulpride
Dotarizine
Deramciclane
Esmirtazapine
Nandrolone decanoate
Cinitapride
Lurasidone
Serotonin
Perospirone
Amperozide
Butriptyline
Cannabidiol
Brexpiprazole
Dosulepin
Etoperidone
Lorpiprazole
Blonanserin
Zotepine
Pipamperone
Setiptiline
Dihydroergocornine
Gilteritinib
Sarpogrelate
Eplivanserin
Ketanserin
Nelotanserin
Ritanserin
Tiapride
Dihydroergocristine
2,5-Dimethoxy-4-ethylthioamphetamine
N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine
Medical Cannabis
5-methoxy-N,N-dimethyltryptamine
Nabiximols
Aripiprazole lauroxil
Volinanserin
Diseases
GWAS
Cardiac hypertrophy (
21348951
)
Femur bone mineral density x serum urate levels interaction (
34046847
)
Parkinson disease and lewy body pathology (
25663231
)
Serum 25-Hydroxyvitamin D levels (
29325163
)
Sjögren's syndrome (
28076899
)
Subcutaneous adipose tissue (
22589738
)
Novel Interacting Genes
6 novel interacting genes:
CTSG
DACH1
DIRAS3
PCDH9
RFXAP
SUGT1
Interacting Genes
19 interacting genes:
ANKS1B
ARF1
ARF6
DLG1
DLG4
EIF3F
GLUL
GNA11
GNAI1
GNAQ
JAK2
MAP1A
MRPL28
NDUFB10
NME3
NTRK3
PON2
PPP5C
RPS6KA3
Entrez ID
3356
HPRD ID
01638
Ensembl ID
ENSG00000102468
Uniprot IDs
A0A7P0PKG8
P28223
PDB IDs
6A93
6A94
6WGT
6WH4
6WHA
7RAN
7VOD
7VOE
7WC4
7WC5
7WC6
7WC7
7WC8
7WC9
8JT8
8UWL
8V6U
8ZMG
Enriched GO Terms of Interacting Partners
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GDP Binding
Postsynaptic Density Organization
G Protein Activity
Guanyl Nucleotide Binding
G-protein Beta/gamma-subunit Complex Binding
G Protein-coupled Serotonin Receptor Signaling Pathway
GTPase Activity
Postsynaptic Specialization Organization
GTP Binding
Nucleotide Binding
Heterotrimeric G-protein Complex
Maintenance Of Postsynaptic Density Structure
Neuron Projection Organization
Synapse
Positive Regulation Of Protein Localization
Phospholipase C-activating Serotonin Receptor Signaling Pathway
Regulation Of Platelet Activation
Plasma Membrane
Protein Localization To Synapse
Maintenance Of Postsynaptic Specialization Structure
Regulation Of Biological Quality
Response To Lipid
Synaptic Membrane
Glutamatergic Synapse
Positive Regulation Of Platelet Aggregation
Acetylcholine Receptor Binding
G Protein-coupled Receptor Binding
Phototransduction, Visible Light
Cytosol
Positive Regulation Of Protein Localization To Cell Periphery
Positive Regulation Of MHC Class II Biosynthetic Process
Regulation Of Protein Localization
Protein Localization To Cell Junction
Response To Ketone
Hydrolase Activity
Positive Regulation Of Homotypic Cell-cell Adhesion
Neurotransmitter Receptor Localization To Postsynaptic Specialization Membrane
Cytoplasm
G Protein-coupled Acetylcholine Receptor Signaling Pathway
Postsynaptic Density
Regulation Of Protein Secretion
Detection Of Visible Light
Regulation Of Presynapse Assembly
Regulation Of Presynapse Organization
Cellular Response To PH
Response To Prostaglandin E
Regulation Of Receptor-mediated Endocytosis
Entrainment Of Circadian Clock
Enzyme Regulator Activity
Regulation Of Cytoskeleton Organization
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