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CASR
Description
calcium sensing receptor
Image
GO Annotations
Cellular Component
Plasma Membrane
Cell Surface
Membrane
Basolateral Plasma Membrane
Apical Plasma Membrane
Axon
Presynaptic Membrane
Neuronal Cell Body
Axon Terminus
Glutamatergic Synapse
Molecular Function
G Protein-coupled Receptor Activity
Integrin Binding
Calcium Ion Binding
Protein Binding
Amino Acid Binding
Protein Kinase Binding
Identical Protein Binding
Protein Homodimerization Activity
Transmembrane Transporter Binding
Metal Ion Binding
Biological Process
Ossification
Response To Ischemia
Detection Of Calcium Ion
Intracellular Calcium Ion Homeostasis
Signal Transduction
G Protein-coupled Receptor Signaling Pathway
Adenylate Cyclase-activating G Protein-coupled Receptor Signaling Pathway
Adenylate Cyclase-inhibiting G Protein-coupled Receptor Signaling Pathway
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
JNK Cascade
Chemosensory Behavior
Positive Regulation Of Cell Population Proliferation
Anatomical Structure Morphogenesis
Response To Metal Ion
Positive Regulation Of Gene Expression
Positive Regulation Of Insulin Secretion
Bile Acid Secretion
Cellular Response To Hepatocyte Growth Factor Stimulus
Vasodilation
Positive Regulation Of Vasoconstriction
Branching Morphogenesis Of An Epithelial Tube
Positive Regulation Of Positive Chemotaxis
Response To Calcium Ion
Regulation Of Calcium Ion Transport
Fat Pad Development
Positive Regulation Of ERK1 And ERK2 Cascade
Cellular Response To Vitamin D
Cellular Response To Glucose Stimulus
Cellular Response To Low-density Lipoprotein Particle Stimulus
Cellular Response To Hypoxia
Response To Fibroblast Growth Factor
Positive Regulation Of Calcium Ion Import
Regulation Of Presynaptic Membrane Potential
Adenylate Cyclase-activating G Protein-coupled CAMP Receptor Signaling Pathway
Positive Regulation Of NLRP3 Inflammasome Complex Assembly
Cellular Response To Peptide
Chloride Transmembrane Transport
Pathways
G alpha (q) signalling events
G alpha (i) signalling events
Class C/3 (Metabotropic glutamate/pheromone receptors)
Drugs
Spermine
Neomycin
Cinacalcet
Ronacaleret
NPS-2143
Calcium citrate
Calcium Phosphate
Etelcalcetide
Calcium phosphate dihydrate
Diseases
Bartter syndrome
GWAS
Calcium levels (
20661308
20705733
24068962
29403010
25886283
25972035
)
Cardiac Troponin-T levels (
23247143
)
Chronic widespread musculoskeletal pain (
33331911
)
Clinical laboratory measurements (
27897004
)
Eosinophil count (
32888494
)
Eosinophil percentage of white cells (
32888494
)
Kidney stones (
26272126
)
Metabolite levels (
31628463
)
Phosphorus levels (
20558539
)
Psoriasis (
25854761
)
QT interval (
29874175
)
Serum parathyroid hormone levels (
27927781
)
Type 2 diabetes (
30718926
32499647
)
Novel Interacting Genes
2 novel interacting genes:
CD200
TCF4
Interacting Genes
11 interacting genes:
FLNA
GRM1
HIF1A
NOTCH1
PI4K2B
PRKCA
PRKCB
PRKCG
RNF19A
STAMBP
VHL
Entrez ID
846
HPRD ID
03122
Ensembl ID
ENSG00000036828
Uniprot IDs
P41180
PDB IDs
5FBH
5FBK
5K5S
5K5T
7DTT
7DTU
7DTV
7DTW
7E6T
7E6U
7M3E
7M3F
7M3G
7M3J
7SIL
7SIM
7SIN
8SZF
8SZG
8SZH
8SZI
8WPG
8WPU
9ASB
9AVG
9AVL
9AXF
9AYF
9C1P
9C2F
9J7I
Enriched GO Terms of Interacting Partners
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Calcium,diacylglycerol-dependent Serine/threonine Kinase Activity
Diacylglycerol-dependent Serine/threonine Kinase Activity
Histone H3T6 Kinase Activity
Negative Regulation Of Apoptotic Process
Regulation Of Intracellular Signal Transduction
Negative Regulation Of Programmed Cell Death
Regulation Of Secretion By Cell
Regulation Of Secretion
Protein Kinase C Signaling
Positive Regulation Of Neural Precursor Cell Proliferation
Regulation Of Exocytosis
Regulation Of Protein Transport
Regulation Of Cell Communication
Regulation Of Signaling
Synaptic Signaling Via Neuropeptide
Regulation Of Apoptotic Process
Regulation Of Establishment Of Protein Localization
Positive Regulation Of Protein Transport
Transcription Regulator Activator Activity
Mitotic Nuclear Membrane Disassembly
Regulation Of Programmed Cell Death
Positive Regulation Of Insulin Secretion
Regulation Of Protein Secretion
Regulation Of Neural Precursor Cell Proliferation
Regulation Of Signal Transduction
Regulation Of Transport
Positive Regulation Of Vascular Endothelial Growth Factor Receptor Signaling Pathway
Membrane Disassembly
Nuclear Membrane Disassembly
Positive Regulation Of Establishment Of Protein Localization
Positive Regulation Of Peptide Hormone Secretion
Regulation Of Cell Population Proliferation
Positive Regulation Of Peptide Secretion
Regulation Of Blood Vessel Endothelial Cell Migration
Calyx Of Held
Phospholipase C-activating G Protein-coupled Receptor Signaling Pathway
Regulation Of Regulated Secretory Pathway
Positive Regulation Of Cell Communication
Positive Regulation Of Signaling
Cellular Response To Hypoxia
Glandular Epithelial Cell Differentiation
Cellular Response To Decreased Oxygen Levels
Positive Regulation Of Protein Secretion
Positive Regulation Of Hormone Secretion
Enzyme Binding
Plasma Membrane
Positive Regulation Of Neuroblast Proliferation
Negative Regulation Of Biomineral Tissue Development
Presynaptic Cytosol
Cellular Response To Oxygen Levels
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